This literature may be useful in answering questions about instrumentation, validation, compaction, tableting, granulation, optimization, etc.

 

Abel JT. Computer system validation:  Questions for the audit. Pharm Eng, 9/10:50-59, 1993

Achanta AS, Adusumilli P, James KW. Endpoint determination and its relevance to physicochemical characteristics of solid dosage forms. Drug Dev Ind Pharm, 23(6):539-546, 1997

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Akande OF, Ford JL, Rubinstein MH. Effect of dwell times on the pre-and main compression of a 1:1 paracetamol: microcrystalline cellulose. J Pharm Pharmacol, 47:1102, 1995

Akande OF, Rubinstein MH, Ford JL. Examination of the compaction properties of a 1:1 acetaminophen: microcrystalline cellulose mixture using precompression and main compression. J Pharm Sci, 86(8), 1997

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Alderborn G. Granule properties of importance to tableting. Acta Pharm Seuc, 25:229-238, 1988

Alderborn G, Duberg M, Nystrom C. Studies on direct compression of tablets. X. Measurement of tablet surface area by permeametry. Powder Technol, 41:49, 1985

Alkan MH, Yuksel A. Granulation in a fluidized bed II.  effect of binder amount on the final granule. Drug Dev Ind Pharm, 12:1529, 1986

Altaf SA, Hoag SW. The effect of tablet machine elasticity on the work of compaction. AAPS Meeting, November, 1993

Altaf SA, Hoag SW. Deformation of the Stokes B2 rotary tablet press:  Quantitation and influence on tablet compaction. J Pharm Sci, 84(3):337-343, 1995

Altaf SA, Hoag SW, Ayres JW`. Bead compacts. I. Effect of compression on maintenance of polymer coat integrity in multilayered bead formulations. Drug Dev Ind Pharm, 24(8):737-746, 1998

Anderson VL, MacLean RA. Design of experiments: A realistic approach. Marcel Dekker Inc., New York, 1974

Andersson J, Lindberg NO. Diosna P25 high-speed mixer equipped with instruments for measuring the rate of rotation of the main impeller motor shaft. Drug Dev Ind Pharm, 9:1495-1505, 1983

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Armstrong NA. Time-dependent factors involved in powder compression and tablet manufacture. Int J Pharm, 49: 1-13, 1989

Armstrong NA. Considerations of compression speed in tablet manufacture. Pharm Tech, 9: 106-116, 1990

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Armstrong NA, Blundell LP. The effect of machine speed on the compaction of some directly compressible tablet diluents. Pharmacol, 37:28P, 1985

Armstrong NA, et al. . Pharmacol, 35:320-321, 1983

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Armstrong NA, Govan IT. Changes in punch velocity profiles during the compaction process. J Pharm Pharmacol, 41S:123P, 1989

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Armstrong NA, Palfrey LP. The effect of machine speed on consolidation of four directly compressible tablet diluents. J Pharm Pharmacol, 41:149-151, 1989

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Asgharnejad M, Storey D. Application of a compaction simulator to the design of a high-dose tablet formulation. Part I. Drug Dev Ind Pharm, 22(9&10):967-975, 1996

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Baert L, Remon JP, Knight P. A comparison between the extrusion forces and sphere quality of a gravity feed extruder and a ram feed extruder. Int J Pharm, 86:1187-192, 1992

Baichwal AR, Augsburger LL. Development and validation of a modified annular shear cell (MASC) to study fictional products of lubricants. Int J Pharm, 26:191-196, 1985

Baie SB, Newton JM, Podczeck F. The characterization of the mechanical properties of pharmaceutical materials. Eur J Pharm Biopharm, 42:138-141, 1996

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Barnett ME, Muller FX, Venkatesh GM. Characterization of the tableting properties of four drug substances using a compaction simulator and Hiestand indices of tableting performance. AAPS Meeting, November, 1998

Barnett ME, Muller FX, Venkatesh GM. Characterization of the tableting properties of four drug substances using a compaction simulator and Hiestand's indices of tableting performance. AAPS Meeting, November, 1998

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Bassam F, et al. Young's modulus of powders used as pharmaceutical excipients. Int J Pharm, 64 55, 1990

Bateman SD. A Comparative Investigation of Compression Simulators. Ph. D. Thesis, Liverpool Polytechnic, 1988

Bateman SD. High speed compression simulators in tabletting research. Pharm J, 240:632-633, 1988

Bateman SD, et al. A comparative investigation of compression simulators. Int J Pharm, 49:209-212, 1989

Bateman SD, Rubinstein MH, Thacker HS. Properties of paracetamol tablets produced using high precompression pressures. J Pharm Pharmacol, 41S:32P, 1989

Bateman SD, Rubinstein MH, Thacker HS. Pre - and main compression in tableting. Pharm Tech Int, 2:30-36, 1990

Bateman SD, Rubinstein MH, Wright P. The effect of compression speed on the properties of ibuprofen tablets. J Pharm Pharmacol, 39:66P, 1987

Becker D, Rigassi T, Bauer-Brandl A. Effectiveness of binders in wet granulation: a comparison using model formulations of different tabletability. Drug Dev Ind Pharm, 23(8):791-808, 1997

Benkerrour L, et al. Granule and tablet formulae study by principal component analysis. Int J Pharm, 19:27-34, 1984

Berchielli AM, Johnson BA, Dumont F. An at-line method for endpoint determination of film coating process that contain active drug substances. AAPS Meeting, November, 1997

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Beten DB, Yuksel N, Baykara T. The changes in the mechanic properties of a direct tableting agent microcrystalline cellulose by precompression. Drug Dev Ind Pharm, 20:2333, 1994

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Bier HP, Leuenberger H, Sucker H. Determination of the uncritical quantity of granulating liquid by power measurements on planetary mixers. Pharm Ind, 4:375-380, 1979

Billardon P, Ozil P, Guyot JC. Planning experiments using an instrumented tablet machine in formulation. Drug Dev Ind Pharm, 13(14):2477-2493, 1987

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Blaey CJ de, Polderman J. Compression of Pharmaceuticals II. Registration and determination of force-displacement curves using a small digital computer. Pharm Weekblad, 106:57-65, 1971

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Bouckaert S, et al. Optimization of a granulation procedure for a hydrophilic matrix tablet using experimental design. Drug Dev Ind Pharm, 22(4):321-327, 1996

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Box GEP, et al. Statistics for Experimenters. Wiley, New York, , 1978

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Brittain HG, et al. Physical characterization of pharmaceutical solids. Pharm Res, 8:963, 1991

Britten JR, Barnett MI, Armstrong NA. Studies on powder plug formation using a simulated capsule filling machine. J Pharm Pharmacol, 48:249-254, 1996

Britten JR, Barnett MI, Armstrong NA. Studies on powder plug formation using a simulated capsule filling machine. J Pharm Pharmacol, 48:249-254, 1996

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Cabelka TD, et al. Comparison of high-shear, low-shear, and fluid bed granulation of vitamin C a strain gaged torque sensor. AAPS Meeting, November, 1992

Carless JE, Leigh S. Compression Characteristics of Powders: Radial die wall pressure transmission and density changes. J Pharm Pharmacol, 26:289-297, 1974

Carlson GT, et al. Design, fabrication and start-up of a laboratory scale compaction simulator. AAPS Meeting, November, 1998

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Carstensen JT. Theory of wet granulation. TechSource Conf, , 1988

Carstensen JT, et al. Correlation between hysteresis loop areas of lower punch and of die pressures versus upper punch pressures. Drug Dev Ind Pharm, 7(5), 645-648, 1981

Çelik M. Computer Aided Studies of the Tablet Compression Process. Ph. D. Thesis, Leicester Polytechnic, 1984

Çelik M. Overview of compaction data analysis techniques. Drug Dev Ind Pharm, 18:767-810, 1992

Çelik M. The past, present, and future of tableting technology. Drug Dev Ind Pharm, 22(1):1-10, 1996

Çelik M, Aulton M. The viscoelastic deformation of some tableting materials as assessed by indentation rheology. Drug Dev Ind Pharm, 22(1):67-75, 1996

Çelik M, Driscoll CE. An overview of the effects of some physico-chemical and mechanical characteristics of particulates on the compaction and post-compaction properties of compacts. Drug Dev Ind Pharm, 19:2119-2141, 1993

Çelik M, et al. Compaction simulator studies of a new drug substance: Effect of particle size and shape, and its binary mixtures with microcrystalline cellulose. Pharm Dev Tech, 1:119-126, 1996

Çelik M, Lordi NG. The pharmaceutical compaction research laboratory and information center. Pharm Tech, 3:112-116, 1991

Çelik M, Marshall K. Use of a compaction simulator system in tableting research.  Part 1:  Introduction to and initial experiments with the system. Drug Dev Ind Pharm, 15:759-800, 5, 1989

Çelik M, Mollan MJ. Minutes of pharmaceutical compaction laboratory consortium meeting. Pharm Tech Int Conf, May 18, 1990

Çelik M, Mollan MJ, Chang N. The reworkability of microcrystalline formulations. PharmTech Conf, Bologna, Italy, 1:239-262, 1991

Çelik M, Okutgen E. A feasibility study for the development of a prospective compaction functionality test and the establishment of a compaction data bank. Drug Dev Ind Pharm, 19:2309-2334, 1993

Çelik M, Ruegger CE. An Overview of Tableting Technology, Part I:  Tablet presses and instrumentation. Pharm Tech Suppl - TabGran Yearbook, 20-39, 1996

Çelik M, Travers DN. The use of elastic recovery index as a criterion of compactional behaviour of some direct compression bases. Drug Dev Ind Pharm, 11:299-314, 1985

Çelik M, Travers DN, Butlery TC. Computer logged changes of strain movements in compacts of direct compression bases and granules produced by wet massing techniques. Pharm Tech Int Conf, 80-89, 1983

Chalmers AA, Elworthy PH. Oxytetracycline tablet formulations: the effect of wet mixing time, particle size and batch variation on granule and tablet properties. J Pharm Pharmacol, 82:239, 1976

Chamberlain R. Computer systems validation for the pharmaceutical and medical device industries. Alaren, Libertyville, IL, 1991

Chang RK, Lai JW. Analysis of content uniformity data using a scatter plot and the tolerance ellipse. Pharm Tech, 5:60-66, 1994

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Chatlapalli R, Rohera BD. Optimization of formulation and process variables for pelletization by extrusion and spheronization using response surface design. AAPS Meeting, November, 1997

Chen Y, et al. Prediction of tablet drug content and hardness using the artificial neural network (ANN) and near-infrared spectroscopy (NIRS). AAPS Meeting, November, 1998

Chen Y, et al. Comparison of artificial neural network (ANN) software in the design of controlled-release formulations. AAPS Meeting, November, 1998

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Chilamkurti RN, Rhodes CT, Schwartz JB. Compression properties of formulations containing matrix and drug. Pharm Acta Helv, 58:146-152, 1983

Chilamkurti RN, Schwartz JB, Rhodes CT. Effect of addition of a soluble and an insoluble drug on the disintegration of tablets made of microcrystalline cellulose and dicalcium phosphate dehydrate. Pharm Acta Helv, 58:251-255, 1983

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Chowhan ZT. Development of a new drug substance into a compacted tablet. Pharm Tech, 9:58-67, 1992

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CSUG. Compaction Simulator Users Group Meeting  - Standards. http://www.bath.ac.uk/, March 23rd, 1996

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Heda PK, Muller FX, Augsburger LL. Capsule filling machine simulation.  I.  Low-force powder compression physics relevant to plug formation. Pharm Dev Tech, 4(2):209-219, 1999

Heda PK, Muteba K, Augsburger LL. Comparison of the formulation requirements of dosator and dosing disc automatic capsule filling machines. AAPS Meeting, November, 1998

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